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1-{2-oxo-3-[(1R)-1-(1H-pyrrol-2-yl)ethyl]-2H-indol-5-yl}urea
- Development stage
- Unknown
- Modality
- Small Molecules
01
Overview
This compound is a synthetic small molecule belonging to the indole and urea chemical classes. It is an experimental molecule, not approved for clinical use, and has primarily been studied as a research tool. The structure features an indolinone core with a pyrrole substituent and a urea moiety. Literature links this scaffold to the inhibition of protein kinases, specifically phosphoinositide-dependent kinase 1 (PDK1), suggesting its mechanism of action may involve kinase inhibition[8]. However, there are no approved therapeutic indications or marketed products containing this compound[3][4][8].
- Other names
- (2-oxo-3-((1R)-1-(1H-pyrrol-2-yl)ethyl)-2H-indol-5-yl)urea{2-oxo-3-[(1R)-1-(1H-pyrrol-2-yI)ethyl]-2H-indol–5-yI}urea1-(2-OXO–3–((IR)-l-(IH-PYRROL–Z-YL)ETHYL)—ZH—INDOL—S-YL)UREA
02
Targets
PDK (Pyruvate dehydrogenase kinase isoform 1)
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